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iimveliso

Vorolazan Intermediate 5 – (2-fluorophenyl) – 1 – [(pyridin-3-yl) sulfonyl] – 1H-pyrrol-3-formaldehyde CAS No. 881677-11-8

Inkcazelo emfutshane:

Elinye Igama:TAK438
Ifomula yemolekyuli:I-C16H11FN2O3S
Ubunzima beMolekyuli:330.333


Iinkcukacha zeMveliso

Iithegi zeMveliso

Inkcazo

I-Vorolazan ePhakathi iyisithako esibalulekileyo kwi-synthesis ye-Vorolazan, i-blocker enamandla kwaye ekhethiweyo ye-potassium-competitive acid esetyenziselwa ukunyanga isifo se-reflux ye-gastroesophageal (GERD) kunye nezinye izifo ezinxulumene ne-asidi.Le khompawundi ephakathi yinxalenye ephambili kwimveliso yeVorolazan kwaye ibalulekile kwishishini lamayeza.

I-Vorolazan intermediates inobunyulu obuphezulu kunye nesakhiwo sekhemikhali esichanekileyo, esenza ukuba zilungele i-R & D kunye nemveliso enkulu.Iimveliso zethu zithatha amanyathelo angqongqo olawulo lomgangatho ukuqinisekisa ukungaguquguquki kunye nokuthembeka kwazo, zizenze zilungele abavelisi bamayeza kunye nabaphandi.

Le ngqungquthela ixabiswa kakhulu kumashishini amayeza njengoko idlala indima ephambili kwi-synthesis yeVorolazan, ichiza eliphumelelayo lokunyanga izifo ezinxulumene ne-asidi.Njengoko iVorolazan iqhubeka nokuqaphela ukusebenza kwayo ekulawuleni isifo se-reflux ye-gastroesophageal kunye neemeko ezinxulumene nazo, imfuno ye-Vorolazan intermediates iyanda.

Khetha Thina

I-JDK iphethe izixhobo zokuvelisa iklasi yokuqala kunye nezixhobo zokulawula uMgangatho, oqinisekisa ukunikezelwa okuzinzile kwe-API intermediates.Iqela lobuchwephesha liqinisekisa iR&D ngemveliso.Ngokuchasene nazo zombini, sikhangela i-CMO kunye ne-CDMO kwimarike yasekhaya neyamanye amazwe.


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